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- CAS Registry #:1260907-17-2
- Formula:C22H22ClN5O2
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| Description: |
I-BET-762 is a small molecule inhibitor of the BET family of bromodomaincontaining proteins. It has been shown to bind to the acetylated lysine recognition motifs on the bromodomain of BET proteins. This binding prevents the interaction of between BET p |
| Synonym(s): |
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide |
| Solubility: |
Soluble in Water |
| Storage / Stability: |
Store at or below –20°C. Solid form is stable at least 12 months from date of receipt, when stored as directed. Do not store aqueous solutions for more than one day. |
| Reference(s): |
Nicodeme E, et al. Nature. 2010 Dec 23;468 (7327):1119-23. |
| Scientific Category: |
Bromodomain(s) |
| Product Type: |
Inhibitors / Activators |
